{"id":5323,"date":"2021-06-18T09:01:03","date_gmt":"2021-06-18T16:01:03","guid":{"rendered":"https:\/\/fuentesfidedignas.com.mx\/?p=5323"},"modified":"2021-06-18T09:01:04","modified_gmt":"2021-06-18T16:01:04","slug":"identifican-moleculas-que-frenan-la-entrada-del-coronavirus-a-las-celulas","status":"publish","type":"post","link":"https:\/\/fuentesfidedignas.com.mx\/index.php\/2021\/06\/18\/identifican-moleculas-que-frenan-la-entrada-del-coronavirus-a-las-celulas\/","title":{"rendered":"Identifican mol\u00e9culas que frenan la entrada del coronavirus a las c\u00e9lulas"},"content":{"rendered":"\n<p><strong><em>La investigaci\u00f3n permitir\u00e1 desarrollo de f\u00e1rmacos antivirales, as\u00ed como la creaci\u00f3n de un tratamiento preventivo contra el coronavirus.<\/em><\/strong><\/p>\n\n\n\n<p>Ciudad de M\u00e9xico.- Cient\u00edficos espa\u00f1oles han logrado identificar las mol\u00e9culas que consiguen frenar la entrada del coronavirus en las c\u00e9lulas, un descubrimiento que podr\u00eda abrir la puerta para desarrollar f\u00e1rmacos antivirales eficaces contra el SARS-CoV-2 responsable del Covid-19.<\/p>\n\n\n\n<p>Lo han logrado investigadores del Consejo Superior de Investigaciones Cient\u00edficas (CSIC), que han conseguido identificar distintos compuestos moleculares que impiden esa entrada del coronavirus en las c\u00e9lulas.<\/p>\n\n\n\n<p>Seg\u00fan explic\u00f3 el CSIC en una nota de prensa difundida este viernes, esos compuestos moleculares consiguen inhibir la interacci\u00f3n que se produce entre la prote\u00edna de la esp\u00edcula del virus y los receptores celulares.<\/p>\n\n\n\n<p>Estas mol\u00e9culas act\u00faan en etapas muy tempranas del ciclo replicativo del virus, por lo que podr\u00edan impedir la hiperactivaci\u00f3n del sistema inmunol\u00f3gico que acaba desencadenando la \u201ctormenta de citoquinas\u201d caracter\u00edstica durante el agravamiento del Covid-19.<\/p>\n\n\n\n<p>Los compuestos identificados como inhibidores de la entrada del virus son mol\u00e9culas propias del grupo de investigaci\u00f3n que lidera Mar\u00eda Jes\u00fas P\u00e9rez P\u00e9rez, investigadora del CSIC en el Instituto de Qu\u00edmica M\u00e9dica (IQM-CSIC).<\/p>\n\n\n\n<p>\u201cEmpleando el s\u00edmil de la puerta, persiguen bloquear la puerta principal por la que el virus accede al interior celular. De este modo, proteger\u00edan a las c\u00e9lulas de la infecci\u00f3n viral\u201d, explic\u00f3 Mar\u00eda Jes\u00fas P\u00e9rez, que lidera el proyecto junto con Sonsoles Mart\u00edn Santamar\u00eda, del Centro de Investigaciones Biol\u00f3gicas Margarita Salas (CIB-CSIC), Ron Geller, del Instituto de Biolog\u00eda Integrativa y de Sistemas, un centro mixto del CSIC y la Universidad de Valencia (este de Espa\u00f1a) y Alberto Marina y Vicente Rubio, del Instituto de Biomedicina de Valencia (IBV-CSIC).<\/p>\n\n\n\n<p>Los investigadores ensayaron los f\u00e1rmacos usando \u201cpseudopart\u00edculas\u201d virales con la prote\u00edna de la esp\u00edcula del virus, y a continuaci\u00f3n analizaron su capacidad para interferir entre la uni\u00f3n de la prote\u00edna de la esp\u00edcula con el receptor celular y la posterior infecci\u00f3n.<\/p>\n\n\n\n<p>\u201cHemos logrado la inhibici\u00f3n de la entrada del virus a concentraciones bajas sin que se genere toxicidad en las c\u00e9lulas hu\u00e9sped; esto genera un amplio \u00edndice de selectividad, un par\u00e1metro que mide la diferencia en concentraciones entre la actividad antiviral y la toxicidad frente a c\u00e9lulas no infectadas; se trata de un factor importante a la hora de desarrollar f\u00e1rmacos antivirales\u201d, se\u00f1al\u00f3 la investigadora del CSIC.<\/p>\n\n\n\n<p>Los compuestos identificados act\u00faan en etapas muy tempranas del ciclo replicativo viral, y al impedir la replicaci\u00f3n del virus en la c\u00e9lula, podr\u00edan evitar los efectos de la \u201ctormenta de citoquinas\u201d que se produce en los casos m\u00e1s graves.<\/p>\n\n\n\n<p>\u201cIncluso se podr\u00eda valorar su uso como tratamiento preventivo de la infecci\u00f3n. A partir de ahora, se inicia un largo camino que incluye su estudio precl\u00ednico y su evaluaci\u00f3n de eficacia en un modelo animal\u201d, inform\u00f3 la investigadora.<\/p>\n\n\n\n<p>El proyecto que ha permitido este descubrimiento ha sido financiado por la Plataforma Salud Global del CSIC y el Fondo Supera Covid-19 que pusieron en marcha la Conferencia de Rectores de Universidades Espa\u00f1olas, el Consejo Superior de Investigaciones Cient\u00edficas (CSIC) y el Banco Santander.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>La investigaci\u00f3n permitir\u00e1 desarrollo de f\u00e1rmacos antivirales, as\u00ed como la creaci\u00f3n de un tratamiento preventivo contra el coronavirus. Ciudad de M\u00e9xico.- Cient\u00edficos espa\u00f1oles han logrado identificar las mol\u00e9culas que consiguen frenar la entrada del coronavirus en las c\u00e9lulas, un descubrimiento que podr\u00eda abrir la puerta para desarrollar f\u00e1rmacos antivirales eficaces contra el SARS-CoV-2 responsable del [&hellip;]<\/p>\n","protected":false},"author":22,"featured_media":5324,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"tdm_status":"","tdm_grid_status":"","footnotes":""},"categories":[39],"tags":[332,59,416],"class_list":{"0":"post-5323","1":"post","2":"type-post","3":"status-publish","4":"format-standard","5":"has-post-thumbnail","7":"category-noticias-nacionales","8":"tag-coronavirus","9":"tag-covid-19","10":"tag-sars-cov-2"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.3 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Identifican mol\u00e9culas que frenan la entrada del coronavirus a las c\u00e9lulas - Fuentes Fidedignas<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/fuentesfidedignas.com.mx\/index.php\/2021\/06\/18\/identifican-moleculas-que-frenan-la-entrada-del-coronavirus-a-las-celulas\/\" \/>\n<meta property=\"og:locale\" content=\"es_MX\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Identifican mol\u00e9culas que frenan la entrada del coronavirus a las c\u00e9lulas - Fuentes Fidedignas\" \/>\n<meta property=\"og:description\" content=\"La investigaci\u00f3n permitir\u00e1 desarrollo de f\u00e1rmacos antivirales, as\u00ed como la creaci\u00f3n de un tratamiento preventivo contra el coronavirus. 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